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Paolo De Caprariis

Pubblicazioni

2021

Massa, A.; Di Mola, A.; De Caprariis, P.(2021). Enantioselective synthesis of isoindolinones
EP 3292102 Università di Salerno
ID:208463 Brevetto (285)

2020

Caputo, L.; Piccialli, I.; Ciccone, R.; de Caprariis, P.; Massa, A.; De Feo, V.; Pannaccione, A.(2020). Lavender and coriander essential oils and their main component linalool exert a protective effect against amyloid-β neurotoxicity. PHYTOTHERAPY RESEARCH. Vol. 2020. Pag.1-8 ISSN:0951-418X.
ID:186400 Articolo in rivista (262)

2017

DE CAPRARIIS, Paolo; DI MOLA, Antonia; Massa, Antonio(2017). Isoindolinoni, procedimenti per la produzione di loro derivati chirali e impiego di questi ultimi
102015902348105 Università di Salerno
ID:170680 Brevetto (285)
De Capraris, Paolo; Di Mola, Antonia; Massa, Antonio(2017). Isoindolinoni, procedimenti per la produzione di loro derivati chirali e impiego di questi ultimi" (Isoindolinones, methods for the production of chiral derivatives and their applications)
IT 1429728 Autori, Unisa
ID:69964 Brevetto (285)
DI MOLA, Antonia; Massa, Antonio; DE FEO, Vincenzo; Basile, Anna; Pascale, Maria; Aquino, Rita Patrizia; DE CAPRARIIS, Paolo(2017). Effect of citral and citral related compounds on viability of pancreatic and human B-lymphoma cell lines. MEDICINAL CHEMISTRY RESEARCH. Vol. 26. Pag.631-639 ISSN:1054-2523.
ID:107986 Articolo in rivista (262)

2016

DI MOLA, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; DE CAPRARIIS, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna(2016). Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 26. Pag.5284-5289 ISSN:0960-894X.
ID:98639 Articolo in rivista (262)
DI MOLA, Antonia; Caruso, Tonino; DE CAPRARIIS, Paolo; Massa, Antonio(2016). Reaction of benzal bromides in water/dioxane system for easy access to benzaldehydes and 2-formylbenzonitriles (2-cyanobenzaldehydes). ARKIVOC. Vol. 4. Pag.9-20 ISSN:1551-7004.
ID:94467 Articolo in rivista (262)

2015

DI MOLA, Antonia; Tiffner, Maximilliam; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; DE CAPRARIIS, Paolo; Waser, Mario; Massa, Antonio(2015). Bifunctional Phase Transfer Catalysis in the Asymmetric Synthesis of Biologically Active Isoindolinones. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY. Vol. 11. Pag.2591-2599 ISSN:1860-5397.
ID:79748 Articolo in rivista (262)
Versione online

2014

Peduto, Antonella; Bruno, Ferdinando; Dehm, Friedrike; Krauth, Verena; DE CAPRARIIS, Paolo; Weinigel, Christina; Barz, Dagmar; Massa, Antonio; De Rosa, Mario; Werz, Oliver; Filosa, Rosanna(2014). Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 81. Pag.492-498 ISSN:0223-5234.
ID:98351 Articolo in rivista (262)
L., Di Matteo; O., Christodoulakis; R., Filosa; DE CAPRARIIS, Paolo; DI MOLA, Antonia; Vasca, Ermanno; Massa, Antonio(2014). New chelating agents for Cu(II), Fe(III), Al(III) and Zn(II) based on beta-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone. JOURNAL OF COORDINATION CHEMISTRY. Vol. 67. Pag.2217-2228 ISSN:0095-8972.
ID:2742 Articolo in rivista (262)

2012

Antonia Di, Mola; Gianluca, Croce; Vijaykumar, More; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio(2012). Active methylene compounds in a very effective approach to 3-substitutedisobenzofuranones through tandem aldol/lactonization reactions. TETRAHEDRON. Vol. 68. Pag.6146-6151 ISSN:0040-4020.
ID:44899 Articolo in rivista (262)
Peduto, Antonella; Rosanna, Filosa; DE CAPRARIIS, Paolo; DE FEO, Vincenzo; Shiyou, Li; Ping, Wang; DE MARTINO, Laura(2012). 1-Methoxy-Canthin-6-One and Related b-Carbolines: From Natural Compound to Synthesis and Biological Activities. In Atta-ur-Rahman STUDIES IN NATURAL PRODUCTS CHEMISTRY Pag.81-104 , . ISBN:9780444518545
ID:53964 Contributo in volume (Capitolo o Saggio) (268)
Carmen, Petronzi; Selene, Collarile; Gianluca, Croce; Filosa, Rosanna; DE CAPRARIIS, Paolo; Peduto, Antonella; Palombi, Laura; Valentina, Intintoli; Antonia Di, Mola; Massa, Antonio(2012). Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 27. Pag.5357-5365 ISSN:1434-193X.
ID:49355 Articolo in rivista (262)

2011

Vijaykumar, More; DI MOLA, Antonia; Milena, Perillo; DE CAPRARIIS, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio(2011). The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones. SYNTHESIS. Vol. 18. Pag.3027-3031 ISSN:0039-7881.
ID:36625 Articolo in rivista (262)
More, VIJAYKUMAR SHIUDAS; DE CAPRARIIS, Paolo; Massa, Antonio(2011). The Aldol Addition of 1,3-Dicarbonyl Compounds to 2-Cyanobenzaldehyde in the Synthesis of Novel 3-Substituted Isoindolinones. In: Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS) Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS)
Pesaro October 17-19
In: Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS) Roma Italian Society of Chemistry Pag.45-45
ID:70350 Poster (275)
Petronzi, Carmen; R., Filosa; Peduto, Antonella; Monti, Maria Chiara; Margarucci, Luigi; Massa, Antonio; Ercolino, Simona Francesca; Bizzarro, Valentina; Parente, Luca; Riccio, Raffaele; DE CAPRARIIS, Paolo(2011). Structure-Based Design, Synthesis and Preliminary Anti-inflammatory Activity of Bolinaquinone Analogues. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 46. Pag.488-496 ISSN:0223-5234.
ID:35771 Articolo in rivista (262)
Peduto, Antonella; More, VIJAYKUMAR SHIUDAS; DE CAPRARIIS, Paolo; Festa, Michela; Capasso, Anna; Piacente, Sonia; DE MARTINO, Laura; DE FEO, Vincenzo; Rosanna, Filosa(2011). Synthesis and Cytotoxic Activity of New beta-carboline Derivatives. MINI-REVIEWS IN MEDICINAL CHEMISTRY. Vol. 11. Pag.486-491 ISSN:1389-5575.
ID:37467 Articolo in rivista (262)
Vijaykumar, More; DI MOLA, Antonia; Gianluca, Croce; Tedesco, Consiglia; Carmen, Petronzi; Peduto, Antonella; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio(2011). Multi-component, regio-selective aldol addition of b-ketoesters to aldehydes: scope and applications. ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 9. Pag.8483-8488 ISSN:1477-0520.
ID:37604 Articolo in rivista (262)
Peduto, Antonella; Massa, Antonio; DI MOLA, Antonia; DE CAPRARIIS, Paolo; Paolo La, Colla; Roberta, Loddo; Sergio, Altamura; Giovanni, Maga; Filosa, Rosanna(2011). 2,3-Dihydro-1,2-Diphenyl-substituted 4HPyridinone Derivatives as New Anti Flaviviridae Inhibitors. CHEMICAL BIOLOGY & DRUG DESIGN. Vol. 77. Pag.441-449 ISSN:1747-0285.
ID:36631 Articolo in rivista (262)
Versione online

2010

Sellitto, Grazia; Aurora, Faruolo; DE CAPRARIIS, Paolo; Sergio, Altamura; Giacomo, Paonessa; Gennaro, Ciliberto(2010). Synthesis and anti-hepatitis C virus activity of novel ethyl 1H-indole-3-carboxylates in vitro.. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 18. Pag.6143-6148 ISSN:1464-3391.
ID:43782 Articolo in rivista (262)
Cioffi, Giuseppina; Pesca Maria, Sabina; DE CAPRARIIS, Paolo; Braca, Alessandra; Severino, Lorella; DE TOMMASI, Nunziatina(2010). Phenolic compounds in olive oil and olive pomace from Cilento (Campania, Italy) and their antioxidant activity.. FOOD CHEMISTRY. Vol. 121. Pag.105-111 ISSN:0308-8146.
ID:36515 Articolo in rivista (262)

2009

Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo(2009). A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride. SYNTHESIS. Vol. 4. Pag.643-649 ISSN:0039-7881.
ID:31069 Articolo in rivista (262)
Filosa, Rosanna; Peduto, Antonella; DI MICCO, Simone; DE CAPRARIIS, Paolo; Festa, Michela; Petrella, Antonello; Giovanni, Capranico; Bifulco, Giuseppe(2009). Molecular modelling studies, synthesis and biological activity of a series of novelbisnaphthalimides and their development as new DNA topoisomeraseII inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 17. Pag.13-24 ISSN:0968-0896.
ID:36641 Articolo in rivista (262)
Filosa, Rosanna; M., Carmela Fulco; Maura, Marinozzi; Nicola, Giacchè; Antonio, Macchiarulo; Peduto, Antonella; Massa, Antonio; DE CAPRARIIS, Paolo; Christian, Thomsen; Claus T., Christoffersen; Roberto, Pellicciari(2009). Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-basedx-acidic amino acids as glutamate receptors ligands. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 17. Pag.242-250 ISSN:0968-0896.
ID:36642 Articolo in rivista (262)

2008

RUOCCO L., A; Viggiano, D; Pignatelli, M; Iannaccone, T; RIMOLI M., G; Melisi, D; Curcio, A; DE LUCIA, S; Carboni, E; CARNEVALE U. A., Gironi; DE CAPRARIIS, Paolo; Sadile, A. G.(2008). Galactosilated dopamine increases attention without reducing activity in C57BL/6 mice. BEHAVIOURAL BRAIN RESEARCH. Vol. 187. Pag.449-454 ISSN:0166-4328.
ID:20889 Articolo in rivista (262)
Cioffi, Giuseppina; DAL PIAZ, Fabrizio; Vassallo, A; Venturella, F; DE CAPRARIIS, Paolo; DE SIMONE, F; DE TOMMASI, Nunziatina(2008). Antiproliferative Oleanane Saponins from Meryta denhamii.. JOURNAL OF NATURAL PRODUCTS. Vol. 71. Pag.1000-1004 ISSN:0163-3864.
ID:22264 Articolo in rivista (262)

2007

Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina(2007). Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives. CURRENT DRUG DELIVERY. Vol. 4. Pag.205-210 ISSN:1567-2018.
ID:36645 Articolo in rivista (262)
Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B.(2007). Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate.. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 336. Pag.133-139 ISSN:0378-5173.
ID:20879 Articolo in rivista (262)

2006

Cioffi, Giuseppina; DAL PIAZ, Fabrizio; DE CAPRARIIS, Paolo; P, ; Sanogo, R; Marzocco, Stefania; Autore, Giuseppina; DE TOMMASI, Nunziatina(2006). Antiproliferative triterpene saponins from Entada africana. JOURNAL OF NATURAL PRODUCTS. Vol. 69. Pag.1323-1329 ISSN:0163-3864.
ID:13966 Articolo in rivista (262)
Melisi, D; Secondo, A; Montoro, Paola; Piacente, Sonia; Rimoli, Mg; Minale, M; DE CAPRARIIS, Paolo; Annunziato, L.(2006). Galactosyl Derivatives of L-Arginine and D-Arginine: Synthesis, Stability, Cell Permeation, and Nitric Oxide Production in Pituitary GH3 Cells. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 49. Pag.4826-4833 ISSN:0022-2623.
ID:14147 Articolo in rivista (262)
Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi(2006). Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery. AAPS PHARMSCITECH. Vol. 7. Pag.E1-E9 ISSN:1530-9932.
ID:36644 Articolo in rivista (262)

2004

Pau, A; Asproni, B; Boatto, G; GRELLA G., E; DE CAPRARIIS, Paolo; Costantino, L; Pinna, G. A.(2004). Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives.. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 21. Pag.545-552 ISSN:0928-0987.
ID:20880 Articolo in rivista (262)

2003

Boatto, G; Nieddu, M; FAEDDA M., V; DE CAPRARIIS, Paolo(2003). Enantiomeric separation by HPLC of 1,4-dihydropyridines with vancomycin as chiral sector. CHIRALITY. Vol. 15. Pag.494-497 ISSN:0899-0042.
ID:20881 Articolo in rivista (262)
Saturnino, Carmela; M., Buonerba; G., Boatto; Pascale, Maria; Moltedo, Ornella; L., DE NAPOLI; D., Montesarchio; J. C., Lancelot; DE CAPRARIIS, Paolo(2003). Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent.. CHEMICAL & PHARMACEUTICAL BULLETIN. Vol. 51. Pag.971-974 ISSN:0009-2363.
ID:3425 Articolo in rivista (262)
Bonina, F; Puglia, C; RIMOLI M., G; Melisi, D; Boatto, G; Neddu, M; Calignano, A; LA RANA, G; DE CAPRARIIS, Paolo(2003). Glycosyl derivatives of dopamine and l-dopa as Anti-Parkinson prodrugs: Synthesis pharmacological activity and in vitro stability studies. JOURNAL OF DRUG TARGETING. Vol. 11. Pag.25-36 ISSN:1061-186X.
ID:20882 Articolo in rivista (262)

2002

Bonina, F.; Puglia, C.; Ventura, D.; Aquino, Rita Patrizia; Tortora, S.; Sacchi, A.; Saija, A.; Tomaino, A.; Pellegrino, M. L.; DE CAPRARIIS, Paolo(2002). In vitro antioxidant and in vivo photoprotective effects of a lyophilized extract of Capparis spinosa L. buds. JOURNAL OF COSMETIC SCIENCE. Vol. 53. Pag.321-335 ISSN:1525-7886.
ID:4794 Articolo in rivista (262)
F. P., Bonina; M. G., Rimoli; L. A., Vallone; M., Amato; C., Puglia; M., Ricci; DE CAPRARIIS, Paolo; F., Barbato(2002). New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical prperties and skin permeation studies.. JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 91. Pag.171-179 ISSN:0022-3549.
ID:20884 Articolo in rivista (262)
DE CAPRARIIS, Paolo; Giampiero, Boatto; Maria, Nieddu; Mauro, Cataldi; Daniela, Melisi; Salvatore, Amoroso(2002). Separation and analysis of the pharmacologic properties of chiral dihydropyridines: comparative evaluation of optical isomers of amlodipine and lercanidipine.. RAPPORTI ISTISAN. Vol. 2. Pag.5-10 ISSN:1123-3117.
ID:44143 Articolo in rivista (262)
Bonina, F; Puglia, C; RIMOLI M., G; Avallone, L; Abbignente, E; Boatto, G; Neddu, M; Meli, R; Amorena, M; DE CAPRARIIS, Paolo(2002). Synthesis and in vitro chemical and enzymatica stability of glycosil 3'-azido-3'-deoxythymidine derivatives as potential anti-HIV agents. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 16. Pag.167-174 ISSN:0928-0987.
ID:20883 Articolo in rivista (262)

2001

Bonina, F; Puglia, C; Barbuzzi, T; DE CAPRARIIS, Paolo; Palagiano, F; RIMOLI M., G; Saia, A.(2001). In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of chetoprofen, naproxen and diclofenac. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 14. Pag.123-134 ISSN:0928-0987.
ID:20885 Articolo in rivista (262)

2000

DE CAPRARIIS, Paolo(2000). Separation of optical antipodes of calcium antagonist drugs and in vitro and in vivo evaluation of the enantiomer stability and pharmacological activities by biochemical methods.. RAPPORTI ISTISAN. Vol. 00/18. Pag.5-12 ISSN:1123-3117.
ID:44144 Articolo in rivista (262)
F. P., Bonina; L., Arenare; R., Ippolito; G., Boatto; G., Battaglia; V., Bruno; DE CAPRARIIS, Paolo(2000). Synthesis, Pharmacokinetics and anticonvulsant activity of 7 – chlorokynurenic acid prodrugs. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 202. Pag.79-88 ISSN:0378-5173.
ID:20886 Articolo in rivista (262)

1999

Cataldi, M; Taglialatela, M; Palagiano, F; Secondo, A; DE CAPRARIIS, Paolo; Amoroso, S; DI RENZO, G; Annunziata, L.(1999). EFFECTS OF MANIDIPINE AND NITRENDIPINE ENANTHUIOMERS ON THE PALTEAU PHASE OF K+-INDUCED INTRACELLULAR Ca2+ INCREASE IN GH3 CELLS. EUROPEAN JOURNAL OF PHARMACOLOGY. Vol. 376. Pag.169-178 ISSN:0014-2999.
ID:20887 Articolo in rivista (262)
F. P., Bonina; L., Arenare; F., Palagiano; A., Saija; F., Nava; D., Trombetta; DE CAPRARIIS, Paolo(1999). Synthesis, stability, and pharmacological evaluation of nipecotic acid prodrugs. JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 88. Pag.561-567 ISSN:0022-3549.
ID:20888 Articolo in rivista (262)
Rimoli Maria, Grazia; Luigi, Avallone; DE CAPRARIIS, Paolo; Aldo, Galeone; Flavio, Forni; Maria Angela, Vandelli(1999). Synthesis and characterization of poly(dl-lactic acid)-idoxuridine conjugate. JOURNAL OF CONTROLLED RELEASE. Vol. 58. Pag.61-68 ISSN:0168-3659.
ID:43797 Articolo in rivista (262)

1998

DE CAPRARIIS, Paolo; Francesco, Palagiano; Mauro, Cataldi; Maurizio, Taglialatela; Salvatore, Amoroso(1998). Separation of the optical antipodes of calcium antagonists and evaluation of their pharmacological activities.. RAPPORTI ISTISAN. Vol. 98. Pag.5-7 ISSN:1123-3117.
ID:44141 Articolo in rivista (262)
Loredana, Arenare; Rosa, Ippolito; Francesco P., Bonina; Giuseppe, Battaglia; Valeria, Bruno; Ferdinando, Nicoletti; DE CAPRARIIS, Paolo(1998). New prodrugs of 7-chlorokynurenic acid. Synthesis, pharmacokinetics and anticonvulsant activity.. ACTA TECHNOLOGIAE ET LEGIS MEDICAMENTI. Vol. 9. Pag.93-98 ISSN:1121-2098.
ID:44137 Articolo in rivista (262)

1997

Francesco, Palagiano; Francesco Paolo, Bonina; Lucia, Montenegro; Biondi, A.; Ludovico, Sorrentino; Capasso, Anna; DE CAPRARIIS, Paolo(1997). Synthesis, stability, and anticonvulsant activity of two new GABA prodrugs.. PHARMAZIE. Vol. 52. Pag.272-276 ISSN:0031-7144.
ID:44270 Articolo in rivista (262)
Capasso, Anna; Biondi, A.; Francesco, Palagiano; Bonina, F. P.; Montenegro, L.; DE CAPRARIIS, Paolo; Pistorio, E.; Sorrentino, L.(1997). Anticonvulsive activity of a new GABA mimetic drug.. EUROPEAN NEUROPSYCHOPHARMACOLOGY. Vol. 7. Pag.57-63 ISSN:0924-977X.
ID:44576 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; Barbato, ; Maria Immacolata La, Rotonda; Fabiana, Quaglia; Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo(1997). In vitro and in vivo evaluation of terpenoid esters of indomethacin as dermal prodrugs. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 149. Pag.171-182 ISSN:0378-5173.
ID:44252 Articolo in rivista (262)
Maria Grazia, Rimoli; Luigi, Avallone; DE CAPRARIIS, Paolo; Elena, Luraschi; Enrico, Abignente; Walter, Filippelli; Liberato, Berrino; Francesco, Rossi(1997). Research on heterocyclic compounds. XXXVII. Synthesis and antiinflammatory activity of methyl-substituted imidazo[1,2-a]pyrazine derivatives.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 32. Pag.195-203 ISSN:0223-5234.
ID:44263 Articolo in rivista (262)

1996

Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo; Francesco, Palagiano; Capasso, Anna; Ludovico, Sorrentino(1996). Pharmacokinetic and pharmacodynamic profile of triethylene glycol indomethacin ester as a new oral prodrug.. JOURNAL OF CONTROLLED RELEASE. Vol. 41. Pag.187-193 ISSN:0168-3659.
ID:44295 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; DE CAPRARIIS, Paolo; Giuliano, Grandolini; Valeria, Ambrogi; Luana, Perioli; Walter, Filippelli; Giuseppe, Falcone; Francesco, Rossi(1996). Synthesis and SAR study of imidazo[2,1-b]benzothiazole acids and some related compounds with anti-inflammatory and analgesic activities.. IL FARMACO. Vol. 51. Pag.483-491 ISSN:0014-827X.
ID:44287 Articolo in rivista (262)
Francesco, Palagiano; DE CAPRARIIS, Paolo; Francesco Paolo, Bonina; Lucia, Montenegro; Capasso, Anna; Ludovico, Sorrentino(1996). Pharmacokinetic and pharmacodynamic profiles of the trioxyethylene ester of indomethacin as a new oral prodrug. BOLLETTINO CHIMICO FARMACEUTICO. Vol. 135. Pag.89-91 ISSN:0006-6648.
ID:44291 Articolo in rivista (262)
Lucia, Avallone; DE CAPRARIIS, Paolo; Aldo, Galeone; Maria Grazia, Rimoli(1996). 1H and 13C NMR spectra of imidazo[1,2-a]pyrazines.. MAGNETIC RESONANCE IN CHEMISTRY. Vol. 34. Pag.409-414 ISSN:0749-1581.
ID:44440 Articolo in rivista (262)

1995

F. P., Bonina; L., Montenegro; DE CAPRARIIS, Paolo; Francesco, Palagiano; G., Trapani; G., Liso(1995). In vitro and in vivo evaluation of polyoxyethylene indomethacin esters as dermal prodrugs. JOURNAL OF CONTROLLED RELEASE. Vol. 34. Pag.223-232 ISSN:0168-3659.
ID:44580 Articolo in rivista (262)
Antonia, Sacchi; DE CAPRARIIS, Paolo; Luciano, Mayol; Giovanni De, Martino(1995). Synthesis and characterization of 4-hydroxy-3-phenylprolines.. JOURNAL OF HETEROCYCLIC CHEMISTRY. Vol. 32. Pag.1067-1069 ISSN:0022-152X.
ID:44563 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; Elena, Luraschi; DE CAPRARIIS, Paolo; Enrico, Abignente; Michele, D'Amico; Walter, Filippelli; Francesco, Rossi(1995). Research on heterocyclic compounds. XXXIV. Synthesis and SAR study of some imidazo[2,1-b]thiazole carboxylic and acetic acids with antiinflammatory and analgesic activities.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 30. Pag.901-909 ISSN:0223-5234.
ID:44446 Articolo in rivista (262)

1993

Giuliano, Grandolini; Valeria, Ambrogi; Luana, Perioli; DE CAPRARIIS, Paolo; Francesco, Palagiano; Maria Grazia, Rimoli; Enrico, Lampa; Michele, D'Amico(1993). Synthesis and pharmacological activity of imidazo[2,1-b]benzothiazole acids. IL FARMACO. Vol. 48. Pag.31-43 ISSN:0014-827X.
ID:44462 Articolo in rivista (262)

1992

Abignente, E; DE CAPRARIIS, Paolo; Rimoli, Mg; Capasso, F; Autore, Giuseppina(1992). Research on heterocyclic compounds, XXIX. Synthesis and antiinflammatory activity of imidazo[1,2-a]pyrazine derivatives.. IL FARMACO. Vol. 47. Pag.919-930 ISSN:0014-827X.
ID:46998 Articolo in rivista (262)

1991

Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo; E., Bousquet; S., Tirendi(1991). 1-Alkylazacycloalkan-2-one esters as prodrugs of indomethacin forimproved delivery through human skin. PHARMACEUTICS. Vol. 77. Pag.21-29 ISSN:1999-4923.
ID:44498 Articolo in rivista (262)
Enrico, Abignente; Francesca, Arena; DE CAPRARIIS, Paolo; Elena, Luraschi; Antonia, Sacchi; Enrico, Lampa; Libero, Berrino; Donato Donnoli, .(1991). Research on heterocyclic compounds. XXVIII. Imidazo[1,2-c]pyrimidines.. IL FARMACO. Vol. 46. Pag.1099-1110 ISSN:0014-827X.
ID:44469 Articolo in rivista (262)

Articolo in rivista (262)

DI MOLA, Antonia; Tiffner, Maximilliam; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; DE CAPRARIIS, Paolo; Waser, Mario; Massa, Antonio(2015). Bifunctional Phase Transfer Catalysis in the Asymmetric Synthesis of Biologically Active Isoindolinones. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY. Vol. 11. Pag.2591-2599 ISSN:1860-5397.
ID:79748 Articolo in rivista (262)
Versione online
DE CAPRARIIS, Paolo(2000). Separation of optical antipodes of calcium antagonist drugs and in vitro and in vivo evaluation of the enantiomer stability and pharmacological activities by biochemical methods.. RAPPORTI ISTISAN. Vol. 00/18. Pag.5-12 ISSN:1123-3117.
ID:44144 Articolo in rivista (262)
DE CAPRARIIS, Paolo; Giampiero, Boatto; Maria, Nieddu; Mauro, Cataldi; Daniela, Melisi; Salvatore, Amoroso(2002). Separation and analysis of the pharmacologic properties of chiral dihydropyridines: comparative evaluation of optical isomers of amlodipine and lercanidipine.. RAPPORTI ISTISAN. Vol. 2. Pag.5-10 ISSN:1123-3117.
ID:44143 Articolo in rivista (262)
F. P., Bonina; M. G., Rimoli; L. A., Vallone; M., Amato; C., Puglia; M., Ricci; DE CAPRARIIS, Paolo; F., Barbato(2002). New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical prperties and skin permeation studies.. JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 91. Pag.171-179 ISSN:0022-3549.
ID:20884 Articolo in rivista (262)
Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi(2006). Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery. AAPS PHARMSCITECH. Vol. 7. Pag.E1-E9 ISSN:1530-9932.
ID:36644 Articolo in rivista (262)
DI MOLA, Antonia; Massa, Antonio; DE FEO, Vincenzo; Basile, Anna; Pascale, Maria; Aquino, Rita Patrizia; DE CAPRARIIS, Paolo(2017). Effect of citral and citral related compounds on viability of pancreatic and human B-lymphoma cell lines. MEDICINAL CHEMISTRY RESEARCH. Vol. 26. Pag.631-639 ISSN:1054-2523.
ID:107986 Articolo in rivista (262)
Enrico, Abignente; Francesca, Arena; DE CAPRARIIS, Paolo; Elena, Luraschi; Antonia, Sacchi; Enrico, Lampa; Libero, Berrino; Donato Donnoli, .(1991). Research on heterocyclic compounds. XXVIII. Imidazo[1,2-c]pyrimidines.. IL FARMACO. Vol. 46. Pag.1099-1110 ISSN:0014-827X.
ID:44469 Articolo in rivista (262)
Cataldi, M; Taglialatela, M; Palagiano, F; Secondo, A; DE CAPRARIIS, Paolo; Amoroso, S; DI RENZO, G; Annunziata, L.(1999). EFFECTS OF MANIDIPINE AND NITRENDIPINE ENANTHUIOMERS ON THE PALTEAU PHASE OF K+-INDUCED INTRACELLULAR Ca2+ INCREASE IN GH3 CELLS. EUROPEAN JOURNAL OF PHARMACOLOGY. Vol. 376. Pag.169-178 ISSN:0014-2999.
ID:20887 Articolo in rivista (262)
Francesco, Palagiano; DE CAPRARIIS, Paolo; Francesco Paolo, Bonina; Lucia, Montenegro; Capasso, Anna; Ludovico, Sorrentino(1996). Pharmacokinetic and pharmacodynamic profiles of the trioxyethylene ester of indomethacin as a new oral prodrug. BOLLETTINO CHIMICO FARMACEUTICO. Vol. 135. Pag.89-91 ISSN:0006-6648.
ID:44291 Articolo in rivista (262)
Bonina, F; Puglia, C; Barbuzzi, T; DE CAPRARIIS, Paolo; Palagiano, F; RIMOLI M., G; Saia, A.(2001). In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of chetoprofen, naproxen and diclofenac. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 14. Pag.123-134 ISSN:0928-0987.
ID:20885 Articolo in rivista (262)
Petronzi, Carmen; R., Filosa; Peduto, Antonella; Monti, Maria Chiara; Margarucci, Luigi; Massa, Antonio; Ercolino, Simona Francesca; Bizzarro, Valentina; Parente, Luca; Riccio, Raffaele; DE CAPRARIIS, Paolo(2011). Structure-Based Design, Synthesis and Preliminary Anti-inflammatory Activity of Bolinaquinone Analogues. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 46. Pag.488-496 ISSN:0223-5234.
ID:35771 Articolo in rivista (262)
Francesco, Palagiano; Francesco Paolo, Bonina; Lucia, Montenegro; Biondi, A.; Ludovico, Sorrentino; Capasso, Anna; DE CAPRARIIS, Paolo(1997). Synthesis, stability, and anticonvulsant activity of two new GABA prodrugs.. PHARMAZIE. Vol. 52. Pag.272-276 ISSN:0031-7144.
ID:44270 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; Barbato, ; Maria Immacolata La, Rotonda; Fabiana, Quaglia; Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo(1997). In vitro and in vivo evaluation of terpenoid esters of indomethacin as dermal prodrugs. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 149. Pag.171-182 ISSN:0378-5173.
ID:44252 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; DE CAPRARIIS, Paolo; Giuliano, Grandolini; Valeria, Ambrogi; Luana, Perioli; Walter, Filippelli; Giuseppe, Falcone; Francesco, Rossi(1996). Synthesis and SAR study of imidazo[2,1-b]benzothiazole acids and some related compounds with anti-inflammatory and analgesic activities.. IL FARMACO. Vol. 51. Pag.483-491 ISSN:0014-827X.
ID:44287 Articolo in rivista (262)
Bonina, F.; Puglia, C.; Ventura, D.; Aquino, Rita Patrizia; Tortora, S.; Sacchi, A.; Saija, A.; Tomaino, A.; Pellegrino, M. L.; DE CAPRARIIS, Paolo(2002). In vitro antioxidant and in vivo photoprotective effects of a lyophilized extract of Capparis spinosa L. buds. JOURNAL OF COSMETIC SCIENCE. Vol. 53. Pag.321-335 ISSN:1525-7886.
ID:4794 Articolo in rivista (262)
Pau, A; Asproni, B; Boatto, G; GRELLA G., E; DE CAPRARIIS, Paolo; Costantino, L; Pinna, G. A.(2004). Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives.. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 21. Pag.545-552 ISSN:0928-0987.
ID:20880 Articolo in rivista (262)
Bonina, F; Puglia, C; RIMOLI M., G; Avallone, L; Abbignente, E; Boatto, G; Neddu, M; Meli, R; Amorena, M; DE CAPRARIIS, Paolo(2002). Synthesis and in vitro chemical and enzymatica stability of glycosil 3'-azido-3'-deoxythymidine derivatives as potential anti-HIV agents. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 16. Pag.167-174 ISSN:0928-0987.
ID:20883 Articolo in rivista (262)
DI MOLA, Antonia; Caruso, Tonino; DE CAPRARIIS, Paolo; Massa, Antonio(2016). Reaction of benzal bromides in water/dioxane system for easy access to benzaldehydes and 2-formylbenzonitriles (2-cyanobenzaldehydes). ARKIVOC. Vol. 4. Pag.9-20 ISSN:1551-7004.
ID:94467 Articolo in rivista (262)
Peduto, Antonella; More, VIJAYKUMAR SHIUDAS; DE CAPRARIIS, Paolo; Festa, Michela; Capasso, Anna; Piacente, Sonia; DE MARTINO, Laura; DE FEO, Vincenzo; Rosanna, Filosa(2011). Synthesis and Cytotoxic Activity of New beta-carboline Derivatives. MINI-REVIEWS IN MEDICINAL CHEMISTRY. Vol. 11. Pag.486-491 ISSN:1389-5575.
ID:37467 Articolo in rivista (262)
Giuliano, Grandolini; Valeria, Ambrogi; Luana, Perioli; DE CAPRARIIS, Paolo; Francesco, Palagiano; Maria Grazia, Rimoli; Enrico, Lampa; Michele, D'Amico(1993). Synthesis and pharmacological activity of imidazo[2,1-b]benzothiazole acids. IL FARMACO. Vol. 48. Pag.31-43 ISSN:0014-827X.
ID:44462 Articolo in rivista (262)
Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo; E., Bousquet; S., Tirendi(1991). 1-Alkylazacycloalkan-2-one esters as prodrugs of indomethacin forimproved delivery through human skin. PHARMACEUTICS. Vol. 77. Pag.21-29 ISSN:1999-4923.
ID:44498 Articolo in rivista (262)
DE CAPRARIIS, Paolo; Francesco, Palagiano; Mauro, Cataldi; Maurizio, Taglialatela; Salvatore, Amoroso(1998). Separation of the optical antipodes of calcium antagonists and evaluation of their pharmacological activities.. RAPPORTI ISTISAN. Vol. 98. Pag.5-7 ISSN:1123-3117.
ID:44141 Articolo in rivista (262)
Vijaykumar, More; DI MOLA, Antonia; Milena, Perillo; DE CAPRARIIS, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio(2011). The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones. SYNTHESIS. Vol. 18. Pag.3027-3031 ISSN:0039-7881.
ID:36625 Articolo in rivista (262)
Abignente, E; DE CAPRARIIS, Paolo; Rimoli, Mg; Capasso, F; Autore, Giuseppina(1992). Research on heterocyclic compounds, XXIX. Synthesis and antiinflammatory activity of imidazo[1,2-a]pyrazine derivatives.. IL FARMACO. Vol. 47. Pag.919-930 ISSN:0014-827X.
ID:46998 Articolo in rivista (262)
Cioffi, Giuseppina; DAL PIAZ, Fabrizio; DE CAPRARIIS, Paolo; P, ; Sanogo, R; Marzocco, Stefania; Autore, Giuseppina; DE TOMMASI, Nunziatina(2006). Antiproliferative triterpene saponins from Entada africana. JOURNAL OF NATURAL PRODUCTS. Vol. 69. Pag.1323-1329 ISSN:0163-3864.
ID:13966 Articolo in rivista (262)
L., Di Matteo; O., Christodoulakis; R., Filosa; DE CAPRARIIS, Paolo; DI MOLA, Antonia; Vasca, Ermanno; Massa, Antonio(2014). New chelating agents for Cu(II), Fe(III), Al(III) and Zn(II) based on beta-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone. JOURNAL OF COORDINATION CHEMISTRY. Vol. 67. Pag.2217-2228 ISSN:0095-8972.
ID:2742 Articolo in rivista (262)
Capasso, Anna; Biondi, A.; Francesco, Palagiano; Bonina, F. P.; Montenegro, L.; DE CAPRARIIS, Paolo; Pistorio, E.; Sorrentino, L.(1997). Anticonvulsive activity of a new GABA mimetic drug.. EUROPEAN NEUROPSYCHOPHARMACOLOGY. Vol. 7. Pag.57-63 ISSN:0924-977X.
ID:44576 Articolo in rivista (262)
Filosa, Rosanna; M., Carmela Fulco; Maura, Marinozzi; Nicola, Giacchè; Antonio, Macchiarulo; Peduto, Antonella; Massa, Antonio; DE CAPRARIIS, Paolo; Christian, Thomsen; Claus T., Christoffersen; Roberto, Pellicciari(2009). Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-basedx-acidic amino acids as glutamate receptors ligands. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 17. Pag.242-250 ISSN:0968-0896.
ID:36642 Articolo in rivista (262)
Maria Grazia, Rimoli; Luigi, Avallone; DE CAPRARIIS, Paolo; Elena, Luraschi; Enrico, Abignente; Walter, Filippelli; Liberato, Berrino; Francesco, Rossi(1997). Research on heterocyclic compounds. XXXVII. Synthesis and antiinflammatory activity of methyl-substituted imidazo[1,2-a]pyrazine derivatives.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 32. Pag.195-203 ISSN:0223-5234.
ID:44263 Articolo in rivista (262)
Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B.(2007). Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate.. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 336. Pag.133-139 ISSN:0378-5173.
ID:20879 Articolo in rivista (262)
Loredana, Arenare; Rosa, Ippolito; Francesco P., Bonina; Giuseppe, Battaglia; Valeria, Bruno; Ferdinando, Nicoletti; DE CAPRARIIS, Paolo(1998). New prodrugs of 7-chlorokynurenic acid. Synthesis, pharmacokinetics and anticonvulsant activity.. ACTA TECHNOLOGIAE ET LEGIS MEDICAMENTI. Vol. 9. Pag.93-98 ISSN:1121-2098.
ID:44137 Articolo in rivista (262)
Melisi, D; Secondo, A; Montoro, Paola; Piacente, Sonia; Rimoli, Mg; Minale, M; DE CAPRARIIS, Paolo; Annunziato, L.(2006). Galactosyl Derivatives of L-Arginine and D-Arginine: Synthesis, Stability, Cell Permeation, and Nitric Oxide Production in Pituitary GH3 Cells. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 49. Pag.4826-4833 ISSN:0022-2623.
ID:14147 Articolo in rivista (262)
Peduto, Antonella; Bruno, Ferdinando; Dehm, Friedrike; Krauth, Verena; DE CAPRARIIS, Paolo; Weinigel, Christina; Barz, Dagmar; Massa, Antonio; De Rosa, Mario; Werz, Oliver; Filosa, Rosanna(2014). Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 81. Pag.492-498 ISSN:0223-5234.
ID:98351 Articolo in rivista (262)
DI MOLA, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; DE CAPRARIIS, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna(2016). Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 26. Pag.5284-5289 ISSN:0960-894X.
ID:98639 Articolo in rivista (262)
Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo(2009). A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride. SYNTHESIS. Vol. 4. Pag.643-649 ISSN:0039-7881.
ID:31069 Articolo in rivista (262)
Cioffi, Giuseppina; DAL PIAZ, Fabrizio; Vassallo, A; Venturella, F; DE CAPRARIIS, Paolo; DE SIMONE, F; DE TOMMASI, Nunziatina(2008). Antiproliferative Oleanane Saponins from Meryta denhamii.. JOURNAL OF NATURAL PRODUCTS. Vol. 71. Pag.1000-1004 ISSN:0163-3864.
ID:22264 Articolo in rivista (262)
F. P., Bonina; L., Montenegro; DE CAPRARIIS, Paolo; Francesco, Palagiano; G., Trapani; G., Liso(1995). In vitro and in vivo evaluation of polyoxyethylene indomethacin esters as dermal prodrugs. JOURNAL OF CONTROLLED RELEASE. Vol. 34. Pag.223-232 ISSN:0168-3659.
ID:44580 Articolo in rivista (262)
Boatto, G; Nieddu, M; FAEDDA M., V; DE CAPRARIIS, Paolo(2003). Enantiomeric separation by HPLC of 1,4-dihydropyridines with vancomycin as chiral sector. CHIRALITY. Vol. 15. Pag.494-497 ISSN:0899-0042.
ID:20881 Articolo in rivista (262)
Antonia Di, Mola; Gianluca, Croce; Vijaykumar, More; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio(2012). Active methylene compounds in a very effective approach to 3-substitutedisobenzofuranones through tandem aldol/lactonization reactions. TETRAHEDRON. Vol. 68. Pag.6146-6151 ISSN:0040-4020.
ID:44899 Articolo in rivista (262)
Rimoli Maria, Grazia; Luigi, Avallone; DE CAPRARIIS, Paolo; Aldo, Galeone; Flavio, Forni; Maria Angela, Vandelli(1999). Synthesis and characterization of poly(dl-lactic acid)-idoxuridine conjugate. JOURNAL OF CONTROLLED RELEASE. Vol. 58. Pag.61-68 ISSN:0168-3659.
ID:43797 Articolo in rivista (262)
Bonina, F; Puglia, C; RIMOLI M., G; Melisi, D; Boatto, G; Neddu, M; Calignano, A; LA RANA, G; DE CAPRARIIS, Paolo(2003). Glycosyl derivatives of dopamine and l-dopa as Anti-Parkinson prodrugs: Synthesis pharmacological activity and in vitro stability studies. JOURNAL OF DRUG TARGETING. Vol. 11. Pag.25-36 ISSN:1061-186X.
ID:20882 Articolo in rivista (262)
Peduto, Antonella; Massa, Antonio; DI MOLA, Antonia; DE CAPRARIIS, Paolo; Paolo La, Colla; Roberta, Loddo; Sergio, Altamura; Giovanni, Maga; Filosa, Rosanna(2011). 2,3-Dihydro-1,2-Diphenyl-substituted 4HPyridinone Derivatives as New Anti Flaviviridae Inhibitors. CHEMICAL BIOLOGY & DRUG DESIGN. Vol. 77. Pag.441-449 ISSN:1747-0285.
ID:36631 Articolo in rivista (262)
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Carmen, Petronzi; Selene, Collarile; Gianluca, Croce; Filosa, Rosanna; DE CAPRARIIS, Paolo; Peduto, Antonella; Palombi, Laura; Valentina, Intintoli; Antonia Di, Mola; Massa, Antonio(2012). Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 27. Pag.5357-5365 ISSN:1434-193X.
ID:49355 Articolo in rivista (262)
Antonia, Sacchi; DE CAPRARIIS, Paolo; Luciano, Mayol; Giovanni De, Martino(1995). Synthesis and characterization of 4-hydroxy-3-phenylprolines.. JOURNAL OF HETEROCYCLIC CHEMISTRY. Vol. 32. Pag.1067-1069 ISSN:0022-152X.
ID:44563 Articolo in rivista (262)
Cioffi, Giuseppina; Pesca Maria, Sabina; DE CAPRARIIS, Paolo; Braca, Alessandra; Severino, Lorella; DE TOMMASI, Nunziatina(2010). Phenolic compounds in olive oil and olive pomace from Cilento (Campania, Italy) and their antioxidant activity.. FOOD CHEMISTRY. Vol. 121. Pag.105-111 ISSN:0308-8146.
ID:36515 Articolo in rivista (262)
F. P., Bonina; L., Arenare; R., Ippolito; G., Boatto; G., Battaglia; V., Bruno; DE CAPRARIIS, Paolo(2000). Synthesis, Pharmacokinetics and anticonvulsant activity of 7 – chlorokynurenic acid prodrugs. INTERNATIONAL JOURNAL OF PHARMACEUTICS. Vol. 202. Pag.79-88 ISSN:0378-5173.
ID:20886 Articolo in rivista (262)
RUOCCO L., A; Viggiano, D; Pignatelli, M; Iannaccone, T; RIMOLI M., G; Melisi, D; Curcio, A; DE LUCIA, S; Carboni, E; CARNEVALE U. A., Gironi; DE CAPRARIIS, Paolo; Sadile, A. G.(2008). Galactosilated dopamine increases attention without reducing activity in C57BL/6 mice. BEHAVIOURAL BRAIN RESEARCH. Vol. 187. Pag.449-454 ISSN:0166-4328.
ID:20889 Articolo in rivista (262)
F. P., Bonina; L., Arenare; F., Palagiano; A., Saija; F., Nava; D., Trombetta; DE CAPRARIIS, Paolo(1999). Synthesis, stability, and pharmacological evaluation of nipecotic acid prodrugs. JOURNAL OF PHARMACEUTICAL SCIENCES. Vol. 88. Pag.561-567 ISSN:0022-3549.
ID:20888 Articolo in rivista (262)
Sellitto, Grazia; Aurora, Faruolo; DE CAPRARIIS, Paolo; Sergio, Altamura; Giacomo, Paonessa; Gennaro, Ciliberto(2010). Synthesis and anti-hepatitis C virus activity of novel ethyl 1H-indole-3-carboxylates in vitro.. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 18. Pag.6143-6148 ISSN:1464-3391.
ID:43782 Articolo in rivista (262)
Francesco Paolo, Bonina; Lucia, Montenegro; DE CAPRARIIS, Paolo; Francesco, Palagiano; Capasso, Anna; Ludovico, Sorrentino(1996). Pharmacokinetic and pharmacodynamic profile of triethylene glycol indomethacin ester as a new oral prodrug.. JOURNAL OF CONTROLLED RELEASE. Vol. 41. Pag.187-193 ISSN:0168-3659.
ID:44295 Articolo in rivista (262)
Lucia, Avallone; DE CAPRARIIS, Paolo; Aldo, Galeone; Maria Grazia, Rimoli(1996). 1H and 13C NMR spectra of imidazo[1,2-a]pyrazines.. MAGNETIC RESONANCE IN CHEMISTRY. Vol. 34. Pag.409-414 ISSN:0749-1581.
ID:44440 Articolo in rivista (262)
Filosa, Rosanna; Peduto, Antonella; DI MICCO, Simone; DE CAPRARIIS, Paolo; Festa, Michela; Petrella, Antonello; Giovanni, Capranico; Bifulco, Giuseppe(2009). Molecular modelling studies, synthesis and biological activity of a series of novelbisnaphthalimides and their development as new DNA topoisomeraseII inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 17. Pag.13-24 ISSN:0968-0896.
ID:36641 Articolo in rivista (262)
Saturnino, Carmela; M., Buonerba; G., Boatto; Pascale, Maria; Moltedo, Ornella; L., DE NAPOLI; D., Montesarchio; J. C., Lancelot; DE CAPRARIIS, Paolo(2003). Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent.. CHEMICAL & PHARMACEUTICAL BULLETIN. Vol. 51. Pag.971-974 ISSN:0009-2363.
ID:3425 Articolo in rivista (262)
Vijaykumar, More; DI MOLA, Antonia; Gianluca, Croce; Tedesco, Consiglia; Carmen, Petronzi; Peduto, Antonella; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio(2011). Multi-component, regio-selective aldol addition of b-ketoesters to aldehydes: scope and applications. ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 9. Pag.8483-8488 ISSN:1477-0520.
ID:37604 Articolo in rivista (262)
Caputo, L.; Piccialli, I.; Ciccone, R.; de Caprariis, P.; Massa, A.; De Feo, V.; Pannaccione, A.(2020). Lavender and coriander essential oils and their main component linalool exert a protective effect against amyloid-β neurotoxicity. PHYTOTHERAPY RESEARCH. Vol. 2020. Pag.1-8 ISSN:0951-418X.
ID:186400 Articolo in rivista (262)
Francesco, Palagiano; Loredana, Arenare; Elena, Luraschi; DE CAPRARIIS, Paolo; Enrico, Abignente; Michele, D'Amico; Walter, Filippelli; Francesco, Rossi(1995). Research on heterocyclic compounds. XXXIV. Synthesis and SAR study of some imidazo[2,1-b]thiazole carboxylic and acetic acids with antiinflammatory and analgesic activities.. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 30. Pag.901-909 ISSN:0223-5234.
ID:44446 Articolo in rivista (262)
Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina(2007). Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives. CURRENT DRUG DELIVERY. Vol. 4. Pag.205-210 ISSN:1567-2018.
ID:36645 Articolo in rivista (262)

Brevetto (285)

DE CAPRARIIS, Paolo; DI MOLA, Antonia; Massa, Antonio(2017). Isoindolinoni, procedimenti per la produzione di loro derivati chirali e impiego di questi ultimi
102015902348105 Università di Salerno
ID:170680 Brevetto (285)
Massa, A.; Di Mola, A.; De Caprariis, P.(2021). Enantioselective synthesis of isoindolinones
EP 3292102 Università di Salerno
ID:208463 Brevetto (285)
De Capraris, Paolo; Di Mola, Antonia; Massa, Antonio(2017). Isoindolinoni, procedimenti per la produzione di loro derivati chirali e impiego di questi ultimi" (Isoindolinones, methods for the production of chiral derivatives and their applications)
IT 1429728 Autori, Unisa
ID:69964 Brevetto (285)

Contributo in volume (Capitolo o Saggio) (268)

Peduto, Antonella; Rosanna, Filosa; DE CAPRARIIS, Paolo; DE FEO, Vincenzo; Shiyou, Li; Ping, Wang; DE MARTINO, Laura(2012). 1-Methoxy-Canthin-6-One and Related b-Carbolines: From Natural Compound to Synthesis and Biological Activities. In Atta-ur-Rahman STUDIES IN NATURAL PRODUCTS CHEMISTRY Pag.81-104 , . ISBN:9780444518545
ID:53964 Contributo in volume (Capitolo o Saggio) (268)

Poster (275)

More, VIJAYKUMAR SHIUDAS; DE CAPRARIIS, Paolo; Massa, Antonio(2011). The Aldol Addition of 1,3-Dicarbonyl Compounds to 2-Cyanobenzaldehyde in the Synthesis of Novel 3-Substituted Isoindolinones. In: Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS) Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS)
Pesaro October 17-19
In: Proceedings of the 11th Sigma-Aldrich Young Chemists Symposium (SAYCS) Roma Italian Society of Chemistry Pag.45-45
ID:70350 Poster (275)